Description of the drug
Pharmacokinetics:
- Complete absorption of yohimbine in the digestive tract occurs after 15–30 minutes after administration
- The highest level of concentration in the blood is observed after 50–70 minutes
- Yohimbine distributes fairly evenly in tissues, and after 15 minutes overcomes the barrier between the blood and the nervous system, entering the cerebrospinal fluid
- About 82% of the drug is protein bound and only about 18% of the extract enters the plasma and brain tissue
- Delivers in about 5 hours
Pharmacodynamics:
- Stimulates sympathetic impulses of the central nervous system
- Releases norepinephrine from nerve endings
- Stabilizes sexual activity
- The extract is non-toxic and does not affect sperm
- Has a beneficial effect on the psycho-emotional background
- Helps relieve feelings of discomfort, stiffness and fear during sexual intercourse
- Activates the process of reducing subcutaneous adipose tissue
Composition of 1 tablet of yohimbine
Active substance | Yohimbine hydrochloride 5 mg |
Additional substances | Gum arabic |
Lactose | |
Corn starch | |
Sucrose | |
Stearic acid | |
Talc |
Release form. Price. Release and storage conditions:
- The release form is predominantly yellowish tablets with a dosage of 5 mg or white bitter powder
- Sold by prescription from your doctor
- Stored in a dry and dark place, out of reach of children, at an air temperature not exceeding 26 °C
- Shelf life – 36 months from the date of production
- Price – 250–350 rub.
Indications for use. Contraindications. Overdose
Indications for use:
- Recommended for use by men who have low sexual activity and potential
- Calms the mental and emotional background
- Helps overcome psychogenic impotence
- Is a preventive measure and generally improves men’s health.
- Used for fat burning purposes
Yohimbine should be taken for:
- Psychogenic impotence
- Strong physical and psycho-emotional stress
- Functional impotence
- Low libido
- Erectile dysfunction
- As a preventive measure, for men over 50 years of age
- Congestion in the prostate
- Atony of the bladder
Contraindications
Despite the fact that yohimbine is a plant alkaloid, it has its contraindications. People with the following diseases should limit their intake of yohimbine:
- Liver or kidney failure
- Peptic ulcer of the stomach or duodenum
- Cardiac ischemia
- Hypertension and hypotension
- Severe nervous excitability
- Excessive anxiety and depression
- If you have insulin-dependent diabetes mellitus
- Insomnia and psychological illnesses
- For atherosclerosis and hyperthyroidism
Overdose
Symptoms of overdose occur approximately 25–35 minutes after ingestion:
- General weakness appears
- Impaired memory and coordination of movements
- Severe headaches
- Migraine
- Dizziness, tachycardia
- Feelings of fear and anxiety
- Vomiting and increased sweating
- 4 hours after taking it, severe pain occurs in the heart area, which can last for a long time
To treat yohimbine overdose:
- Use gastric lavage followed by activated charcoal and sodium sulfate
- In severe cases of poisoning, use 0.1–0.2 mg of clonidine once, and 0.1 mg at intervals every 60 minutes until the symptoms of overdose disappear
Yohimbine for weight loss
This drug is used to solve problems with erection, but its other important property is also known - the ability to burn fat. So, yohimbine for weight loss: how to use this remedy correctly, what results can you expect?
Helpful information
Why is yohimbine used for weight loss, what is its mechanism of action? As you know, alpha-adrenergic receptors are present in our body - they block the release of fat from lipocytes.
Fat is most easily deposited in the abdomen and thighs - there is the highest concentration of such receptors. Yohimbine (an alkaloid obtained from the bark of the African yohimbe tree) blocks these receptors, which allows fat to be burned evenly throughout the body.
It is believed that yohimbine is a kind of testosterone booster, and this hormone causes the body to burn fat. The alkaloid enhances thermogenesis (converts fat calories into heat).
Attention!
When using the drug before training, the release of norepinephrine is accelerated, due to which the concentration of fatty acids in the blood increases by 2 times.
Forms of release of the drug: capsules, tablets, tea. Yohimbine hydrochloride for weight loss can be purchased at the pharmacy. Nutritional supplements and teas with this active ingredient are sold on the Internet, as well as in sports nutrition stores and pharmacies (active ingredient content is about 3%).
Dosage
How to take yohimbine for weight loss? The maximum daily dose of yohimbe extract is 2000 mg (1 dose - 1000 mg), the rate of yohimbe hydrochloride is 30 mg (1 dose - 5 mg). Athletes take the drug at the rate of 0.2 mg/1 kg of body weight. Course duration is 2-3 weeks. You can repeat it after 2 months.
When treating impotence, yohimbine is taken with or after meals, while when treating obesity, it is taken on an empty stomach.
The fact is that this alkaloid, in combination with food, promotes the release of insulin, and this leads to fat deposition rather than burning it. The optimal break between food and the drug is 4 hours. During this period, you are allowed to drink water and coffee.
Caffeine is known to enhance the fat-burning effects of yohimbine. Some athletes use caffeine tablets instead of coffee.
Contraindications
Yohimbine cannot be used for weight loss in case of individual intolerance, as well as hypertension, arrhythmia and hypotension.
You should not use the drug in cases of severe vascular atherosclerosis and hyperthyroidism. Yohimbine is not prescribed for increased nervous excitability and mental disorders.
Important!
Contraindications are kidney and liver pathologies, insulin-dependent diabetes mellitus, as well as prostate diseases in the acute phase.
When taking the drug, heart rhythm disturbances and changes in blood pressure may occur. Sometimes you can hear complaints of headaches, redness of the skin, trembling, disruption of the gastrointestinal tract, and insomnia. Men may experience spontaneous erections.
Price
Yohimbe hydrochloride costs 200-250 rubles (50 tablets). The cost of supplements varies from 200 to 2000 rubles (depending on the composition, manufacturer and the number of tablets in the package).
Reviews
Yohimbine is primarily used by athletes for weight loss. If you don't exercise, you may not expect noticeable weight loss.
Source: https://info.cake.dn.ua/johimbin-dlya-pohudeniya/
Side effects and special instructions
Side effects:
- Fluctuations in blood pressure
- Tachycardia
- Excitement
- Insomnia or drowsiness
- Headache
- Dizziness
- Skin redness
Yohimbe extract should not be taken:
- For patients with glaucoma
- Minors
- The drug is not prescribed to women
- If you have a rare form of galactose intolerance
- People prone to sudden changes in blood pressure and tachycardia
- Simultaneously with taking antidepressants, tranquilizers or any other stimulants of the central nervous system
During treatment you should refrain from:
- Taking alcoholic drinks
- Transport management
- Performing work that requires concentration
Doses and method of administration:
- The medicine is prescribed by the attending physician
- Take 5-10 mg with meals, without chewing and with a glass of water.
- Frequency of administration – 1–3 times a day
- The term of treatment is determined by the doctor; if necessary, the course can be repeated, but not earlier than 3 months after the end of the previous one
Drug compatibility:
- Concomitant use of yohimbine and other drugs that affect the psycho-emotional state is contraindicated.
- Yoquinbine can enhance the effect of antidepressants, antihypertensive drugs, alprozalam and increases the risk of side effects
- Taking clondine during treatment with yoquinbine is not advisable, both drugs neutralize each other
Yohimbine for weight loss: how to take, contraindications “The most effective method for losing weight
Yohimbine for weight loss blocks alpha-adrenergic receptors responsible for the process of releasing fat from lipocytes, suitable for men and women.
Yohimbine for weight loss (yohimbine hydrochloride) is a stimulating alkaloid, a specific organic compound containing nitrogen.
On topic: Exercises for losing weight on your legs
It is considered one of the effective drugs in the fight against impotence in men. Due to its stimulating effect, Yohimbine hydrochloride is used not only as an aphrodisiac, but also as an effective means for weight loss.
This feature of Yohimbine is not described in the official instructions for the drug.
The drug is available in the form of capsules or tablets for oral use. For the treatment of impotence in men, Yohimbine hydrochloride is recommended to take 1-2 capsules three times a day.
This dosage is general - in each specific case, the required dosage of the drug is prescribed individually.
Capsules should be taken directly during or before meals.
The main active component in the composition of the drug is an organic extract from the evergreen plant Yohimbe, belonging to the madder family, growing in the regions of Central Africa, which, after assembly, was crushed and dried. For a long period of time, the drug was used exclusively as a libido stimulant in men - thanks to its stimulating properties, Yohimbine effectively fights physiological and psychological impotence in men.
The main principle of action of Yohimbine hydrochloride is to block alpha-adrenergic receptors, which are responsible for blocking the process of fat release from lipocytes.
These alpha-adrenergic receptors contribute to the active accumulation of fat on the body. Yohimbine acts as a powerful fat burner, allowing you to effectively burn fat in all areas of the body. The drug has a stimulating effect on the central nervous system, activating the motor activity of the body and stimulating the process of burning fat.
When using the product exclusively for weight loss, the recommended dosage differs from that specified in the instructions for the drug. It is calculated individually and directly depends on the general state of health and body weight.
Advice!
0.2 mg of Yohimbine hydrochloride is multiplied by one kg of body weight and the daily dose of the drug is obtained. The resulting figure is divided by 3 - this way you can find out the single dose of the medicine.
The tablets are taken orally without chewing.
If, to stimulate libido in men, the drug is recommended to be taken directly during meals, then when using Yohimbine as a fat burner, it should be taken only on an empty stomach.
This recommendation is due to the fact that simultaneous use of the drug and food significantly reduces the effectiveness of the former. Yohimbine for weight loss should be taken 4-5 hours after meals. When combining the drug and sports activities, it is recommended to take a single dose of the drug 1-1.5 hours before training. This will significantly increase its effectiveness.
- The drug is not recommended for use in the presence of arterial hypotension, vascular atherosclerosis, hypertension, arrhythmia, and diabetes mellitus.
- Women with severe kidney and liver dysfunction should avoid using the drug.
- A variety of mental disorders accompanied by increased nervous excitability are a serious contraindication to the use of the drug.
- The supplement should not be used if individual intolerance to the active components included in the medicine is identified.
- The fat burner is not recommended for women during pregnancy and breastfeeding.
- Also contraindicated is age under 16 years.
In most cases, Yohimbine is well tolerated by the body of both women and men. But in extremely rare cases, this organic remedy can cause some side effects, which include:
- When using the medicine, men may experience spontaneous erection.
- Side effects of the medication may include shortness of breath and a sharp increase in blood pressure.
- Various disorders in the functioning of the gastrointestinal tract - stool disorders, nausea, vomiting, discomfort in the abdominal area.
- Nervous system disorders - frequent headaches, dizziness, anxiety, increased excitability, sudden mood swings, sleep disorders.
- As a result of taking Yohimbine, allergic skin reactions may occur, expressed in the form of rash, redness, and itching.
The average cost of Yohimbine hydrochloride can vary from 190 to 1500 rubles. It depends on the manufacturer, the release form and the number of tablets in the package.
Yohimbine has established itself as a safe and effective fat burner that allows you to quickly get rid of extra pounds. But this remedy should not be considered a panacea - to achieve the desired effect, taking Yohimbine should be combined with a properly selected diet and regular exercise.
Source: https://ultrapohudenie.logdown.com/posts/2123520
Analogs
Yohimbine has a considerable number of medicinal analogues, but they all have some differences:
- Eroton. An oral medication prescribed for men with erectile dysfunction. It can be used for a very long time, but has side effects in the form of unstable color vision impairment. Average price – 1150 rub.
- Levitra. Helps enhance the effects of endogenous nitric oxide in the cavernous bodies, enhances blood circulation and increases blood flow. Average price – 2300 rub.
- Viagra. A selective inhibitor of GMP-specific PDE-5, prescribed for low sexual activity in men. Average price – 8100 rub.